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Darunavir�(dá)蘆那�是一�HIV-1蛋白酶抑制劑,用于治療成�HIV-1感染。然而,在此次爆�(fā)�2019-nCoV新型冠狀病毒疫情�,李蘭娟院士�(tuán)�(duì)根據(jù)初步�(cè)��(fā)�(xiàn),達(dá)蘆那韋在300微摩爾濃度下,能顯著抑制新型冠狀病毒�(fù)�,與未用藥物處理組比�,抑制效率高�(dá)280�,因此建議將此藥物列入國(guó)家衛(wèi)健委《新型冠狀病毒感染的肺炎診療方�(試行第六�)�。該藥已用于治療浙江省新型冠狀病毒感染的肺炎患�,下一步計(jì)劃用此藥物替代其他效果欠佳的藥物,故此藥物有望成為抗新型冠狀病毒的明星藥物之一�

百靈威是集研�(fā)、生�(chǎn)、經(jīng)�(yíng)于一體的高科技化學(xué)公司,在歐洲和亞洲的制造基地裝備了500mL-3000L 的反�(yīng)釜,配套形成先�(jìn)的柔性化�(xué)合成系統(tǒng),生�(chǎn)多種藥物合成�(lǐng)域常用產(chǎn)品;為支持廣大藥廠及科研工作者共抗疫�,百靈威人正在加緊生�(chǎn),提��(dá)蘆那�合成所需�(chǎn)��

 

相關(guān)�(chǎn)�

CAS

名稱

貨號(hào)

分子�(jié)�(gòu)�

78-81-9

 

Isobutylamine, 99%

異丁�

124707

67-63-0

Isopropanol, 99.5%, SuperDry, with molecular sieves, J&KSeal

異丙�超干溶劑帶分子篩, J&KSeal

919270

67-63-0

Isopropanol, 99.5%, SuperDry, J&KSeal

異丙�超干溶劑, J&KSeal

971509

98-74-8

4-Nitrobenzenesulfonyl chloride, 99%

4-硝基苯磺酰氯

357341

141-78-6

Ethyl acetate, 99.9%, SuperDry, with molecular sieves, J&KSeal

乙酸乙酯超干溶劑帶分子篩, J&KSeal

920352

76-05-1

Trifluoroacetic acid, 99.9% 

三氟乙酸

101398

76-05-1

Trifluoroacetic acid, 99%

三氟乙酸

252705

1191-99-7

2,3-Dihydrofuran, 99% 

2,3-二氫呋喃

155814

75-09-2

Dichloromethane, 99.9%, SuperDry, with molecular sieves, water≤30 ppm, J&KSeal 

二氯甲烷超干溶劑帶分子篩, water≤30 ppm, J&KSeal

908525

DCM

75-09-2

Dichloromethane, 99.8% 

二氯甲烷

947068

DCM

688-73-3

Tri-n-butyltin hydride, 97%, for synthesis, stabilized with 0.05% BHT 

三丁基氫化錫用于合成含穩(wěn)定劑: 0.05% BHT

929653

 78-67-1

2,2'-Azoisobutyronitrile, 99% 

偶氮二異丁腈

614752

 67-56-1

Methanol, 99.9%, SuperDry, with molecular sieves, water≤30 ppm, J&KSeal

甲醇超干溶劑帶分子篩, water≤30 ppm, J&KSeal

957329

MeOH

67-56-1

Methanol, 99.9%, SuperDry, water≤30 ppm, J&KSeal

甲醇超干溶劑, water≤30 ppm, J&KSeal

980290

MeOH

75-18-3

Dimethyl sulfide, 99%

甲硫�

593537

64-17-5

Ethanol, 99.5%, SuperDry, with molecular sieves, J&KSeal

乙醇超干溶劑帶分子篩, J&KSeal

922424

EtOH

64-17-5

Ethanol, 99.5%, SuperDry, J&KSeal

乙醇超干溶劑, J&KSeal

954068

EtOH

121-44-8

Triethylamine, 99% 

三乙�

432915

75-05-8

Acetonitrile,99.9%, SuperDry, with molecular sieves, J&Kseal

乙腈超干溶劑帶分子篩, J&Kseal

939631

CH3CN

75-05-8

Acetonitrile, 99.9%, SuperDry, water≤30 ppm, J&Kseal

乙腈超干溶劑水含�≤30 ppm, J&Kseal

909376

CH3CN

74124-79-1

N,N'-Disuccinimidyl carbonate, 99%, reagent grade

N.N'-二琥珀酰亞胺基碳酸�試劑�(jí)

992431

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